GR-45809
 | This article is an orphan, as no other articles link to it. Please introduce links to this page from related articles; try the Find link tool for suggestions. (December 2024) |
 | |
| Identifiers | |
|---|---|
| PubChem CID | |
| ChemSpider | |
| Chemical and physical data | |
| Formula | C20H26Cl2N2O3 |
| Molar mass | 413.34 g·mol−1 |
| 3D model (JSmol) | |
| |
GR-45809 is a kappa opioid receptor (KOR) agonist with use in the treatment of pain.[1][2] It was developed over 30 years ago. It has a structure that is similar to ZT-52656A.
References
[edit]- ^ Vecchietti V, Giordani A, Giardina G, Colle R, Clarke GD (January 1991). "(2S)-1-(arylacetyl)-2-(aminomethyl)piperidine derivatives: novel, highly selective kappa opioid analgesics". Journal of Medicinal Chemistry. 34 (1): 397–403. doi:10.1021/jm00105a061. PMID 1846921.
- ^ Scopes DI, Hayes NF, Bays DE, Belton D, Brain J, Brown DS, Judd DB, McElroy AB, Meerholz CA, Naylor A (February 1992). "New kappa-receptor agonists based upon a 2-[(alkylamino)methyl]piperidine nucleus". Journal of Medicinal Chemistry. 35 (3): 490–501. doi:10.1021/jm00081a009. PMID 1310743.
 | This analgesic-related article is a stub. You can help Wikipedia by expanding it. |